Concise synthesis of 6-formylindolo[3,2-b]carbazole (FICZ)

研究成果: Article

2 引用 (Scopus)

抄録

A concise synthesis of 6-formylindolo[3,2-b]carbazole (FICZ), a potent ligand of the aryl hydrocarbon receptor (AhR), has been established. The conjugate addition of the enolate derived from indolylacetate 2 to 2-chloro-3-formylindole 3 was accomplished. The following cyclization reaction under the acidic conditions gave the indolo[3,2-b]carbazole skeleton.

元の言語English
ページ(範囲)1932-1934
ページ数3
ジャーナルChemistry Letters
43
発行部数12
DOI
出版物ステータスPublished - 2014

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Aryl Hydrocarbon Receptors
Cyclization
Ligands
6-formylindolo(3,2-b)carbazole
3-formylindole
indolo(3,2-b)carbazole

ASJC Scopus subject areas

  • Chemistry(all)

これを引用

Concise synthesis of 6-formylindolo[3,2-b]carbazole (FICZ). / Sekine, Daisuke; Okeda, Shota; Hosokawa, Seijiro.

:: Chemistry Letters, 巻 43, 番号 12, 2014, p. 1932-1934.

研究成果: Article

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